{"id":161,"date":"2015-09-10T13:04:03","date_gmt":"2015-09-10T11:04:03","guid":{"rendered":"http:\/\/jcet.eu\/new\/?page_id=161"},"modified":"2023-02-22T16:34:07","modified_gmt":"2023-02-22T15:34:07","slug":"pracownia-analityki-i-farmakokinetyki-jcet","status":"publish","type":"page","link":"https:\/\/jcet.eu\/new\/o-jcet\/laboratoria-jcet\/pracownia-analityki-i-farmakokinetyki-jcet\/","title":{"rendered":"Analityka i Farmakokinetyka"},"content":{"rendered":"<h2><span style=\"color: #ff0000;\"> Pracownia Analityki i Farmakokinetyki (JCET)<\/span><\/h2>\n<p><img decoding=\"async\" class=\"noimage\" src=\"http:\/\/jcet.eu\/images\/paif_03.jpg\" alt=\"Pracownia analityki i farmakokinetyki\" align=\"left\" border=\"0\" \/><\/p>\n<p align=\"justify\">W Pracowni Analityki i Farmakokinetyki prowadzone s\u0105 badania w zakresie opracowywania oraz walidacji\u00a0 nowych metod analitycznych stosowanych do oznaczania st\u0119\u017cenia zwi\u0105zk\u00f3w endo- oraz egzogennych w materiale biologicznym z zastosowaniem techniki wysokosprawnej chromatografii cieczowej w po\u0142\u0105czeniu ze spektrometri\u0105 mas (LC-MS). Prowadzone badania obejmuj\u0105 mi\u0119dzy innymi ocen\u0119 zmian w biosyntezie moleku\u0142 nisko- oraz wysokocz\u0105teczkowych odzwierciedlaj\u0105cych fenotyp \u015br\u00f3db\u0142onka naczyniowego oraz jego dysfunkcj\u0119 w zwierz\u0119cych modelach chor\u00f3b uk\u0142adu sercowo-naczyniowego. W\u015br\u00f3d profilowanych moleku\u0142 znajduj\u0105 si\u0119 wybrane przeka\u017aniki lipidowe, bia\u0142ka specyficzne dla \u015br\u00f3db\u0142onka, metabolity g\u0142\u00f3wnych szlak\u00f3w biochemicznych (m.in.: TCA, glikoliza) oraz aminokwasy. Ponadto, prowadzone s\u0105 badania z zakresu farmakokinetyki, obejmuj\u0105ce wyznaczanie podstawowych parametr\u00f3w farmakokinetycznych oraz ocen\u0105 profilu farmakokinetycznego (ADME) nowych zwi\u0105zk\u00f3w (potencjalnych lek\u00f3w naczynioprotekcyjnych), poszukiwaniem \u015bcie\u017cek ich metabolizmu oraz ocen\u0105 wi\u0105zania z bia\u0142kami krwi. Kierownikiem PAiF jest dr Agnieszka Kij.<\/p>\n<hr \/>\n<p>Najwa\u017cniejsz\u0105 aparatur\u0119 badawcz\u0105 Pracowni Analityki i Farmakokinetyki stanowi\u0105:<\/p>\n<p align=\"justify\"><strong>Wysokosprawny chromatograf cieczowy Ultimate 3000\u00a0<\/strong>(Dionex) sprz\u0119\u017cony ze\u00a0<strong>spektrometrem mas TSQ QuantumUltra\u00a0<\/strong>(Thermo Scientific) typu potr\u00f3jny kwadrupol. Spektrometr mas wyposa\u017cony jest w grzane \u017ar\u00f3d\u0142o jon\u00f3w pracuj\u0105ce w trybie elektrosprej (HESI) oraz chemicznej jonizacji w ci\u015bnieniu atmosferycznym (APCI). Po\u0142\u0105czenie rozdzielenia chromatograficznego analit\u00f3w z zastosowaniem sytemu LC oraz detekcji poprzez zastosowanie tandemowej spektrometrii mas pozwala na opracowanie dok\u0142adnych, czu\u0142ych oraz wysoce specyficznych metod bioanalitycznych do jednoczesnego oznaczania st\u0119\u017cenia wielu moleku\u0142 w jednej pr\u00f3bce.<\/p>\n<p align=\"justify\"><strong>Wysokosprawny chromatograf cieczowy UFLC Nexera <\/strong>(Schimadzu) sprz\u0119\u017cony ze\u00a0<strong>spektrometrem mas Qtrap 5500 <\/strong>(Sciex) typu potr\u00f3jny kwadrupol. Spektrometr mas ponadto wyposa\u017cony jest w pu\u0142apk\u0119 jon\u00f3w pozwalaj\u0105c\u0105 mi\u0119dzy innymi na prowadzenie analiz w trybie MS3 oraz dodatkow\u0105 identyfikacj\u0119 badanych moleku\u0142. Dzi\u0119ki unikatowej konstrukcji analizatora mas urz\u0105dzenie charakteryzuje si\u0119 wysok\u0105 czu\u0142o\u015bci\u0105 i dok\u0142adno\u015bci\u0105 prowadzonych analiz.<\/p>\n<p align=\"justify\"><strong>Elektroforeza kapilarna\u00a0<\/strong>(Beckman Coulter) w po\u0142\u0105czeniu <strong>z detektorem DAD<\/strong>. Programowalny, zautomatyzowany system pozwalaj\u0105cy na rozdzielenie zwi\u0105zk\u00f3w pod wp\u0142ywem przy\u0142o\u017conego wysokiego napi\u0119cia elektrycznego. Aparat umo\u017cliwia jednoczesne przy\u0142o\u017cenie sta\u0142ego lub gradientowego napi\u0119cia, nat\u0119\u017cenia lub mocy ze sta\u0142ym lub gradientowym ci\u015bnieniem lub pr\u00f3\u017cni\u0105. System stosowany jest do oznaczania st\u0119\u017ce\u0144 aktywnych zwi\u0105zk\u00f3w w matrycach biologicznych, oceny wi\u0105zania badanych zwi\u0105zk\u00f3w i lek\u00f3w z bia\u0142kami krwi oraz wyznaczania ich parametr\u00f3w fizykochemicznych takich jak LogP oraz LogD.<\/p>\n<p align=\"justify\"><strong>Chromatograf cieczowy ENO-20 NOx<\/strong> (Eicom) w po\u0142\u0105czeniu<strong> z detektorem UV\/VIS. <\/strong>System ten stanowi analizator metabolit\u00f3w tlenku azotu (NO), takich jak azotyny oraz azotany. Detekcja metabolit\u00f3w NO jest mo\u017cliwa po ich wcze\u015bniejszym rozdzieleniu na kolumnie chromatograficznej, derywatyzacji z u\u017cyciem odczynnikiem Griessa, a nast\u0119pnie detekcji powsta\u0142ych pochodnych diazowych.<\/p>\n<p align=\"justify\"><strong>Potencjostat ROXY<\/strong> (Antec) w po\u0142\u0105czeniu <strong>ze spektrometrem mas<\/strong> <strong>Qtrap 5500 <\/strong>(Sciex). System pozwalaj\u0105cy na symulacje <em>in chemico<\/em> metabolizmu badanych zwi\u0105zk\u00f3w z uwzgl\u0119dnieniem I oraz II fazy metabolizmu mi\u0119dzy innymi w oparciu o reakcj\u0119 utleniania-redukcji, a nast\u0119pnie detekcj\u0119 oraz identyfikacj\u0119 powsta\u0142ych metabolit\u00f3w z zastosowaniem spektrometrii mas.<\/p>\n<style id=\"bwg-style-0\">    #bwg_container1_0 #bwg_container2_0 .bwg-container-0.bwg-standard-thumbnails {      width: 1804px;              justify-content: center;        margin:0 auto !important;              background-color: rgba(255, 255, 255, 0.00);            padding-left: 4px;      padding-top: 4px;      max-width: 100%;            }        #bwg_container1_0 #bwg_container2_0 .bwg-container-0.bwg-standard-thumbnails .bwg-item {    justify-content: flex-start;      max-width: 360px;            width: 360px !important;          }    #bwg_container1_0 #bwg_container2_0 .bwg-container-0.bwg-standard-thumbnails .bwg-item a {       margin-right: 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po\u0142\u0105czeniu<\/p>\n","protected":false},"author":3,"featured_media":0,"parent":149,"menu_order":3,"comment_status":"closed","ping_status":"closed","template":"","meta":{"_acf_changed":false,"footnotes":""},"class_list":["post-161","page","type-page","status-publish","hentry"],"acf":[],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v28.5 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Analityka i Farmakokinetyka &#187; JCET<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/jcet.eu\/new\/o-jcet\/laboratoria-jcet\/pracownia-analityki-i-farmakokinetyki-jcet\/\" \/>\n<meta property=\"og:locale\" content=\"pl_PL\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Analityka i Farmakokinetyka &#187; JCET\" \/>\n<meta property=\"og:description\" content=\"Pracownia Analityki i 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